CBE Research Report Spring 2014 | Page 9

SOLID-STATE NMR CONSTRAINTS ON MOLECULAR ORGANIZATION WITHIN MAX8 DESIGNER PEPTIDE NANOFIBERS Sarah R. Leonard1,2, Maxwell I. Zimmerman1,2, Xiaodong Pang3, Huan-Xiang Zhou3, Anant K. Paravastu1,2 1 Department of Chemical and Biomedical Engineering, Florida State University, 2525 Pottsdamer Street, Tallahassee, FL 32310 USA 2 National High Magnetic Field Laboratory, Florida State University, 1800 E Paul Dirac Dr, Tallahassee, FL 32310 3 Department of Physics and Institute of Molecular Biophysics, Florida State University, Tallahassee, FL 32306 MAX8, a designer peptide known to undergo self-assembly following changes in temperature, pH, and ionic strength, has demonstrated utility for tissue engineering and drug delivery. Here, we report evidence from solid-state NMR spectroscopy that supports the presence of the hypothesized β-hairpin conformation and constrains the arrangement of MAX8 molecules within nanofibers. Specifically, 13C13 C 2-dimensional correlation spectroscopy indicates spatial proximity between V3 and K17 residues, and 13 C-13C dipolar coupling measurements reveal proximity between the V3 and V18 backbone carbonyls. Moreover, isotopic dilution of labeled MAX8 nanofibers did not result in a loss of the 13C-13C dipolar couplings, showing that these couplings are primarily intramolecular. Additional MAX8 samples were synthesized to differentiate between two possible arrangements of MAX8 molecules: 1) the “syn” configuration, with all β-hairpin hinges aligned along the same edge of the β-sheet, and 2) the “anti” configuration, with alternating β-hairpin hinges aligned along opposite edges of the β-sheet. 13C-13C dipolar coupling measurements indicate weak interactions between neighboring V5 backbone carbonyls, consistent with the syn configuration. Intermolecular 15N-13C dipole-dipole couplings indicate spatial proximity between the V5 backbone carbonyl and the V16 backbone nitrogen, also consistent with the syn configuration. A lack of contact between the V3 and T12 residues with 13C-13C 2-dimensional correlation spectroscopy is indicative of a syn-parallel between-sheet conformation with all β-hairpin hinges aligned along the same edge of the stacked β-sheet. Combined, these results led to the development of an all-atom molecular model of MAX8 nanofibers consistent with current NMR experimental constraints. 8|Page